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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T2493 | PD 151746 | Cysteine Protease , Proteasome | |
PD151746 is a calpain inhibitor with a 20-fold selectivity for u-calpain (Ki = 0.26 ± 0.03 μM) over m-calpain (Ki = 5.33 ± 0.77 μM). Its IC50 values are 0.26 ± 0.03 μM (Ki for μ-calpain) and 5.33 ± 0.77 μM (Ki for m-calp... |